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Found 3 of Enz. Inhib. data with enzyme = 'Prokineticin receptor 1' and Substrate = '[125I]MIT-1'
TargetProkineticin receptor 1(Homo sapiens (Human))
University of Ferrara

LigandPNGBDBM26335(3-[2-({5-[(4-ethylphenyl)methyl]-1-[(4-methoxyphen...)
Affinity DataKi:  22nM ΔG°:  -10.9kcal/molepH: 7.4 T: 2°CAssay Description:Nonspecific binding was determined in the presence of 1 uM Bv8. Displacement curves were determined in triplicate. The inhibition constant (Ki) of th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProkineticin receptor 1(Homo sapiens (Human))
University of Ferrara

LigandPNGBDBM26336(6-[(2-aminoethyl)amino]-3-[(4-ethylphenyl)methyl]-...)
Affinity DataKi:  440nM ΔG°:  -9.01kcal/molepH: 7.4 T: 2°CAssay Description:Nonspecific binding was determined in the presence of 1 uM Bv8. Displacement curves were determined in triplicate. The inhibition constant (Ki) of th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProkineticin receptor 1(Homo sapiens (Human))
University of Ferrara

LigandPNGBDBM26337(6-{[2-(4,5-dihydro-1H-imidazol-2-ylamino)ethyl]ami...)
Affinity DataKi:  4.72E+3nM ΔG°:  -7.55kcal/molepH: 7.4 T: 2°CAssay Description:Nonspecific binding was determined in the presence of 1 uM Bv8. Displacement curves were determined in triplicate. The inhibition constant (Ki) of th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed